Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 18:49:24 GMT 2025
by
admin
on
Tue Apr 01 18:49:24 GMT 2025
|
| Protein Type | RECEPTOR |
| Protein Sub Type | TYROSINE KINASE |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
4CH8636GFF
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
|
Preferred Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
P06213
Created by
admin on Tue Apr 01 18:49:24 GMT 2025 , Edited by admin on Tue Apr 01 18:49:24 GMT 2025
|
PRIMARY | |||
|
INSULIN RECEPTOR
Created by
admin on Tue Apr 01 18:49:24 GMT 2025 , Edited by admin on Tue Apr 01 18:49:24 GMT 2025
|
PRIMARY | |||
|
4CH8636GFF
Created by
admin on Tue Apr 01 18:49:24 GMT 2025 , Edited by admin on Tue Apr 01 18:49:24 GMT 2025
|
PRIMARY |
| From | To |
|---|---|
| 1_8 | 1_26 |
| 1_126 | 1_155 |
| 1_159 | 1_182 |
| 1_169 | 1_188 |
| 1_192 | 1_201 |
| 1_196 | 1_207 |
| 1_208 | 1_216 |
| 1_212 | 1_225 |
| 1_228 | 1_237 |
| 1_241 | 1_253 |
| 1_259 | 1_284 |
| 1_266 | 1_274 |
| 1_288 | 1_301 |
| 1_304 | 1_308 |
| 1_312 | 1_333 |
| 1_435 | 1_468 |
| 1_647 | 2_137 |
| 2_63 | 2_72 |
| 1_524 | 3_524 |
| 3_8 | 3_26 |
| 3_126 | 3_155 |
| 3_159 | 3_182 |
| 3_169 | 3_188 |
| 3_192 | 3_201 |
| 3_196 | 3_207 |
| 3_208 | 3_216 |
| 3_212 | 3_225 |
| 3_228 | 3_237 |
| 3_241 | 3_253 |
| 3_259 | 3_284 |
| 3_266 | 3_274 |
| 3_288 | 3_301 |
| 3_304 | 3_308 |
| 3_312 | 3_333 |
| 3_435 | 3_468 |
| 3_647 | 4_137 |
| 4_63 | 4_72 |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_16 |
| N | 1_25 |
| N | 1_78 |
| N | 1_111 |
| N | 1_215 |
| N | 1_255 |
| N | 1_295 |
| N | 1_337 |
| N | 1_397 |
| N | 1_418 |
| N | 1_514 |
| N | 1_606 |
| N | 1_624 |
| N | 1_671 |
| N | 2_7 |
| N | 2_20 |
| N | 2_158 |
| N | 2_171 |
| N | 3_16 |
| N | 3_25 |
| N | 3_78 |
| N | 3_111 |
| N | 3_215 |
| N | 3_255 |
| N | 3_295 |
| N | 3_337 |
| N | 3_397 |
| N | 3_418 |
| N | 3_514 |
| N | 3_606 |
| N | 3_624 |
| N | 3_671 |
| N | 4_7 |
| N | 4_20 |
| N | 4_158 |
| N | 4_171 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
INHIBITOR -> TARGET |
IC50
|
||
|
AGONIST -> TARGET |
|
||
|
INHIBITOR -> TARGET |
INHIBITOR
IC50
|
||
|
INHIBITOR -> TARGET |
Enzymatic Assay
IC50
|
||
|
INHIBITOR -> TARGET |
|
||
|
AGONIST -> TARGET |
IGF-1 activates the insulin receptor at approximately 0.1x the potency of insulin.
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
ALLOSTERIC INHIBITOR
|
||
|
|
AGONIST -> TARGET |
|
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [2_230] [2_237] [2_249] [2_423] [2_427] [2_428] [2_593] [2_599] | TYROSINE O-PHOSPHATE | 2R86C98KDX | |||
| AMINO ACID SUBSTITUTION | [1_373] [1_380] | DEXFOSFOSERINE | VI4F0K069V | |||
| AMINO ACID SUBSTITUTION | [1_374] | TYROSINE O-PHOSPHATE | 2R86C98KDX |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|