U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 02:05:24 GMT 2025
Edited
by admin
on Wed Apr 02 02:05:24 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
51A15DDJ1W
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
G PROTEIN-COUPLED RECEPTOR KINASE (HUMAN GENE GRK5)
Preferred Name English
G PROTEIN-COUPLED RECEPTOR KINASE 5
Common Name English
G PROTEIN-COUPLED RECEPTOR KINASE GRK5
Common Name English
GPRK5
Common Name English
Code System Code Type Description
EC (ENZYME CLASS)
EC 2.7.11.16
Created by admin on Wed Apr 02 02:05:24 GMT 2025 , Edited by admin on Wed Apr 02 02:05:24 GMT 2025
PRIMARY
CAS
1311334-39-0
Created by admin on Wed Apr 02 02:05:24 GMT 2025 , Edited by admin on Wed Apr 02 02:05:24 GMT 2025
ALTERNATIVE
CAS
631087-44-0
Created by admin on Wed Apr 02 02:05:24 GMT 2025 , Edited by admin on Wed Apr 02 02:05:24 GMT 2025
ALTERNATIVE
CAS
942965-22-2
Created by admin on Wed Apr 02 02:05:24 GMT 2025 , Edited by admin on Wed Apr 02 02:05:24 GMT 2025
ALTERNATIVE
CAS
149661-15-4
Created by admin on Wed Apr 02 02:05:24 GMT 2025 , Edited by admin on Wed Apr 02 02:05:24 GMT 2025
ALTERNATIVE
PHAROS
P34947
Created by admin on Wed Apr 02 02:05:24 GMT 2025 , Edited by admin on Wed Apr 02 02:05:24 GMT 2025
PRIMARY
CAS
1310765-12-8
Created by admin on Wed Apr 02 02:05:24 GMT 2025 , Edited by admin on Wed Apr 02 02:05:24 GMT 2025
ALTERNATIVE
CAS
629689-80-1
Created by admin on Wed Apr 02 02:05:24 GMT 2025 , Edited by admin on Wed Apr 02 02:05:24 GMT 2025
ALTERNATIVE
UNIPROT
P34947
Created by admin on Wed Apr 02 02:05:24 GMT 2025 , Edited by admin on Wed Apr 02 02:05:24 GMT 2025
PRIMARY
CAS
405347-82-2
Created by admin on Wed Apr 02 02:05:24 GMT 2025 , Edited by admin on Wed Apr 02 02:05:24 GMT 2025
ALTERNATIVE
CAS
481298-72-0
Created by admin on Wed Apr 02 02:05:24 GMT 2025 , Edited by admin on Wed Apr 02 02:05:24 GMT 2025
PRIMARY
CAS
1311341-01-1
Created by admin on Wed Apr 02 02:05:24 GMT 2025 , Edited by admin on Wed Apr 02 02:05:24 GMT 2025
ALTERNATIVE
FDA UNII
51A15DDJ1W
Created by admin on Wed Apr 02 02:05:24 GMT 2025 , Edited by admin on Wed Apr 02 02:05:24 GMT 2025
PRIMARY
WIKIPEDIA
GRK5
Created by admin on Wed Apr 02 02:05:24 GMT 2025 , Edited by admin on Wed Apr 02 02:05:24 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_484] SERINE DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_579] SERINE DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_485] THREONINE THREONINE PHOSPHATE 3L4WX7B1EI
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER AVERAGE(CALCULATED) CHEMICAL
Molecular Formula CHEMICAL