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Details

Stereochemistry ACHIRAL
Molecular Formula C29H32N6O.C4H4O4.H2O
Molecular Weight 614.6914
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 1
Charge 0

SHOW SMILES / InChI
Structure of GSK-958108 monomaleate monohydrate

SMILES

O.OC(=O)\C=C/C(O)=O.CC1=NC2=CC=CC(N3CCN(CCC4=C5CCC6=C(N=CN6C5=CC=C4C)C(N)=O)CC3)=C2C=C1

InChI

InChIKey=GZKFZADPUZWVEJ-FJOGWHKWSA-N
InChI=1S/C29H32N6O.C4H4O4.H2O/c1-19-6-10-26-22(9-11-27-28(29(30)36)31-18-35(26)27)21(19)12-13-33-14-16-34(17-15-33)25-5-3-4-24-23(25)8-7-20(2)32-24;5-3(6)1-2-4(7)8;/h3-8,10,18H,9,11-17H2,1-2H3,(H2,30,36);1-2H,(H,5,6)(H,7,8);1H2/b;2-1-;

HIDE SMILES / InChI

Molecular Formula C29H32N6O
Molecular Weight 480.604
Charge 0
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Molecular Formula C4H4O4
Molecular Weight 116.0722
Charge 0
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 1
Optical Activity NONE

Molecular Formula H2O
Molecular Weight 18.0153
Charge 0
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Approval Year

Substance Class Chemical
Created
by admin
on Wed Apr 02 19:34:38 GMT 2025
Edited
by admin
on Wed Apr 02 19:34:38 GMT 2025
Record UNII
56SKM4624P
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
GSK-958108 monomaleate monohydrate
Code English
GSK958108 monomaleate monohydrate
Preferred Name English
GSK958108E
Code English
Imidazo[1,5-a]quinoline-3-carboxamide, 4,5-dihydro-7-methyl-6-[2-[4-(2-methyl-5-quinolinyl)-1-piperazinyl]ethyl]-, (2Z)-2-butenedioate, hydrate (1:1:1)
Systematic Name English
Code System Code Type Description
CAS
1173714-19-6
Created by admin on Wed Apr 02 19:34:38 GMT 2025 , Edited by admin on Wed Apr 02 19:34:38 GMT 2025
PRIMARY
PUBCHEM
44138099
Created by admin on Wed Apr 02 19:34:38 GMT 2025 , Edited by admin on Wed Apr 02 19:34:38 GMT 2025
PRIMARY
FDA UNII
56SKM4624P
Created by admin on Wed Apr 02 19:34:38 GMT 2025 , Edited by admin on Wed Apr 02 19:34:38 GMT 2025
PRIMARY
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PARENT -> SALT/SOLVATE
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ACTIVE MOIETY