U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Mon Mar 31 22:26:30 GMT 2025
Edited
by admin
on Mon Mar 31 22:26:30 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
8EJE45ZR0I
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
AXL ONCOGENE
Preferred Name English
TYROSINE-PROTEIN KINASE RECEPTOR UFO
Common Name English
TYROSINE KINASE RECEPTOR UFO (HUMAN GENE AXL)
Common Name English
UFO
Common Name English
Code System Code Type Description
CAS
1432759-18-6
Created by admin on Mon Mar 31 22:26:30 GMT 2025 , Edited by admin on Mon Mar 31 22:26:30 GMT 2025
ALTERNATIVE
WIKIPEDIA
AXL RECEPTOR TYROSINE KINASE
Created by admin on Mon Mar 31 22:26:30 GMT 2025 , Edited by admin on Mon Mar 31 22:26:30 GMT 2025
PRIMARY
CAS
1432761-16-4
Created by admin on Mon Mar 31 22:26:30 GMT 2025 , Edited by admin on Mon Mar 31 22:26:30 GMT 2025
PRIMARY
EC (ENZYME CLASS)
EC 2.7.10.1
Created by admin on Mon Mar 31 22:26:30 GMT 2025 , Edited by admin on Mon Mar 31 22:26:30 GMT 2025
PRIMARY
FDA UNII
8EJE45ZR0I
Created by admin on Mon Mar 31 22:26:30 GMT 2025 , Edited by admin on Mon Mar 31 22:26:30 GMT 2025
PRIMARY
UNIPROT
P30530
Created by admin on Mon Mar 31 22:26:30 GMT 2025 , Edited by admin on Mon Mar 31 22:26:30 GMT 2025
PRIMARY
PHAROS
P30530
Created by admin on Mon Mar 31 22:26:30 GMT 2025 , Edited by admin on Mon Mar 31 22:26:30 GMT 2025
PRIMARY
From To
1_31 1_92
1_135 1_180
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_18
N 1_132
N 1_173
N 1_314
N 1_320
N 1_376
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
LIGAND->TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
LIGAND->TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
CONJUGATED TOXIN->TARGET
LIGAND->TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_678] [1_754] [1_796] [1_841] TYROSINE TYROSINE O-PHOSPHATE 2R86C98KDX
AMINO ACID SUBSTITUTION [1_859] SERINE DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER AVERAGE(CALCULATED) CHEMICAL