U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 03:00:51 GMT 2025
Edited
by admin
on Wed Apr 02 03:00:51 GMT 2025
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
CGS7YUT37M
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
METABOTROPIC GLUTAMATE RECEPTOR 3
Common Name English
GPRC1C
Preferred Name English
MGLUR3
Common Name English
mGlu3 glutamate receptor
Common Name English
Code System Code Type Description
FDA UNII
CGS7YUT37M
Created by admin on Wed Apr 02 03:00:51 GMT 2025 , Edited by admin on Wed Apr 02 03:00:51 GMT 2025
PRIMARY
From To
1_35 1_77
1_218 1_505
1_339 1_351
1_390 1_397
1_487 1_506
1_491 1_509
1_512 1_524
1_527 1_540
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_187
N 1_270
N 1_392
N 1_417
Related Record Type Details
PARTIAL AGONIST->TARGET
Emax = 62
EC50
AGONIST -> TARGET
NEGATIVE ALLOSTERIC MODULATOR (NAM)->TARGET
INHIBITOR -> TARGET
ANTAGONIST
NEGATIVE ALLOSTERIC MODULATOR->TARGET
AGONIST -> TARGET
Ki
INHIBITOR -> TARGET
Functional assay for cAMP formation.
IC50
INHIBITOR -> TARGET
Ki
INHIBITOR -> TARGET
In Rodents
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT CHEMICAL