U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 19:00:10 GMT 2025
Edited
by admin
on Tue Apr 01 19:00:10 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
DRF8ZSM45D
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
AMPK-RELATED PROTEIN KINASE 5
Preferred Name English
NUAK FAMILY SNF1-LIKE KINASE 1
Common Name English
OMPHALOCELE KINASE 1
Common Name English
ARK5
Common Name English
NUAK1
Common Name English
Code System Code Type Description
PHAROS
O60285
Created by admin on Tue Apr 01 19:00:10 GMT 2025 , Edited by admin on Tue Apr 01 19:00:10 GMT 2025
PRIMARY
FDA UNII
DRF8ZSM45D
Created by admin on Tue Apr 01 19:00:10 GMT 2025 , Edited by admin on Tue Apr 01 19:00:10 GMT 2025
PRIMARY
UNIPROT
O60285
Created by admin on Tue Apr 01 19:00:10 GMT 2025 , Edited by admin on Tue Apr 01 19:00:10 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_211] THREONINE PHOSPHATE 3L4WX7B1EI
AMINO ACID SUBSTITUTION [1_22] [1_455] DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_600] DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_1] N-ACETYLMETHIONINE 9J12WX5B6A
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL