U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 19:56:44 GMT 2025
Edited
by admin
on Tue Apr 01 19:56:44 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
EI5D7HW1BA
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
MAPK/ERK KINASE KINASE 1
Preferred Name English
MITOGEN-ACTIVATED PROTEIN KINASE KINASE KINASE 1
Common Name English
MAPKKK1
Common Name English
MEKK1
Common Name English
MEKK
Common Name English
MEK KINASE 1
Common Name English
Code System Code Type Description
PHAROS
Q13233
Created by admin on Tue Apr 01 19:56:44 GMT 2025 , Edited by admin on Tue Apr 01 19:56:44 GMT 2025
PRIMARY
FDA UNII
EI5D7HW1BA
Created by admin on Tue Apr 01 19:56:44 GMT 2025 , Edited by admin on Tue Apr 01 19:56:44 GMT 2025
PRIMARY
WIKIPEDIA
MAP3K1
Created by admin on Tue Apr 01 19:56:44 GMT 2025 , Edited by admin on Tue Apr 01 19:56:44 GMT 2025
PRIMARY
UNIPROT
Q13233
Created by admin on Tue Apr 01 19:56:44 GMT 2025 , Edited by admin on Tue Apr 01 19:56:44 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_20] [1_34] [1_136] [1_153] [1_291] [1_296] [1_299] [1_506] [1_530] [1_922] [1_1017] [1_1042] S DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_1] A N-ACETYLALANINE 26C4VY6Z0M
AMINO ACID SUBSTITUTION [1_284] [1_1399] [1_1411] T THREONINE PHOSPHATE 3L4WX7B1EI
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL
Molecular Formula CHEMICAL