U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 17:04:54 GMT 2025
Edited
by admin
on Tue Apr 01 17:04:54 GMT 2025
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
JHZ3XB1MNK
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
EPITHELIAL DISCOIDIN DOMAIN-CONTAINING RECEPTOR 1
Common Name English
CD167 ANTIGEN-LIKE FAMILY MEMBER A
Preferred Name English
CD167a
Common Name English
DDR1
Common Name English
RTK6
Common Name English
TRKE
Common Name English
PROTEIN-TYROSINE KINASE 3A
Common Name English
PROTEIN-TYROSINE KINASE RTK-6
Common Name English
HGK2
Common Name English
EDDR1
Common Name English
DISCOIDIN RECEPTOR TYROSINE KINASE
Common Name English
PTK3A
Common Name English
TYROSINE-PROTEIN KINASE CAK
Common Name English
Code System Code Type Description
FDA UNII
JHZ3XB1MNK
Created by admin on Tue Apr 01 17:04:54 GMT 2025 , Edited by admin on Tue Apr 01 17:04:54 GMT 2025
PRIMARY
UNIPROT
Q08345
Created by admin on Tue Apr 01 17:04:54 GMT 2025 , Edited by admin on Tue Apr 01 17:04:54 GMT 2025
PRIMARY
From To
1_13 1_167
1_56 1_159
1_285 1_330
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_193
N 1_242
N 1_352
N 1_353
N 1_376
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_466] [1_495] [1_502] [1_722] [1_774] [1_778] [1_779] TYROSINE O-PHOSPHATE 2R86C98KDX
AMINO ACID SUBSTITUTION [1_613] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL
Molecular Formula CHEMICAL