U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 16:52:13 GMT 2025
Edited
by admin
on Tue Apr 01 16:52:13 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
L01TYM08QX
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
FGFR-3
Preferred Name English
FIBROBLAST GROWTH FACTOR RECEPTOR 3
Common Name English
JTK4
Common Name English
FGFR3
Common Name English
Code System Code Type Description
PHAROS
P22607
Created by admin on Tue Apr 01 16:52:13 GMT 2025 , Edited by admin on Tue Apr 01 16:52:13 GMT 2025
PRIMARY
UNIPROT
P22607
Created by admin on Tue Apr 01 16:52:13 GMT 2025 , Edited by admin on Tue Apr 01 16:52:13 GMT 2025
PRIMARY
FDA UNII
L01TYM08QX
Created by admin on Tue Apr 01 16:52:13 GMT 2025 , Edited by admin on Tue Apr 01 16:52:13 GMT 2025
PRIMARY
From To
1_39 1_87
1_154 1_206
1_253 1_317
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_76
N 1_203
N 1_240
N 1_272
N 1_293
N 1_306
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
MUTANT->PARENT
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
DERIVATIVE -> PARENT
CONJUGATED TOXIN->TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
at higher concentrations that were still clinically achievable
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_422] [1_423] DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_625] [1_626] [1_702] [1_738] TYROSINE O-PHOSPHATE 2R86C98KDX
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL
Molecular Formula CHEMICAL