Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 18:47:35 GMT 2025
by
admin
on
Tue Apr 01 18:47:35 GMT 2025
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| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
L5R0QCN8LZ
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| Record Status |
Validated (UNII)
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| Record Version |
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-
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| Code System | Code | Type | Description | ||
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P26358
Created by
admin on Tue Apr 01 18:47:35 GMT 2025 , Edited by admin on Tue Apr 01 18:47:35 GMT 2025
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PRIMARY | |||
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L5R0QCN8LZ
Created by
admin on Tue Apr 01 18:47:35 GMT 2025 , Edited by admin on Tue Apr 01 18:47:35 GMT 2025
|
PRIMARY |
| Linkage Type | Residue Index | |
|---|---|---|
| ZINC FINGER | 1_646 | 1_692 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
Inhibits DNMT1 on a hemimethylated substrate
Ki
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_160] [1_173] [1_188] [1_259] [1_366] [1_749] [1_891] [1_957] [1_961] [1_975] [1_1054] [1_1111] [1_1113] [1_1115] [1_1119] [1_1121] [1_1349] [1_1415] | N<SUP>2</SUP>-ACETYL-L-LYSINE | 7D44E6BN1B |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| Molecular Formula | CHEMICAL |
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| MOL_WEIGHT | CHEMICAL |
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