U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 18:56:38 GMT 2025
Edited
by admin
on Tue Apr 01 18:56:38 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
LR4LA8YD5Z
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
BRD2
Preferred Name English
BROMODOMAIN-CONTAINING PROTEIN 2
Common Name English
RING3
Common Name English
REALLY INTERESTING NEW GENE 3 PROTEIN
Common Name English
KIAA9001
Common Name English
O27.1.1
Common Name English
Code System Code Type Description
UNIPROT
P25440
Created by admin on Tue Apr 01 18:56:38 GMT 2025 , Edited by admin on Tue Apr 01 18:56:38 GMT 2025
PRIMARY
FDA UNII
LR4LA8YD5Z
Created by admin on Tue Apr 01 18:56:38 GMT 2025 , Edited by admin on Tue Apr 01 18:56:38 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
BRD2(BD2) DOMAIN
Kd
INHIBITOR -> TARGET
INHIBITOR -> TARGET
Kd
INHIBITOR -> TARGET
A >250x differential binding preference for BDII over BDI
BINDING
INHIBITOR -> TARGET
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_6] THREONINE PHOSPHATE 3L4WX7B1EI
AMINO ACID SUBSTITUTION [1_1] N-ACETYLMETHIONINE 9J12WX5B6A
AMINO ACID SUBSTITUTION [1_37] [1_298] [1_301] [1_305] [1_633] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL