Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 18:56:38 GMT 2025
by
admin
on
Tue Apr 01 18:56:38 GMT 2025
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
LR4LA8YD5Z
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Preferred Name | English | ||
|
Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
P25440
Created by
admin on Tue Apr 01 18:56:38 GMT 2025 , Edited by admin on Tue Apr 01 18:56:38 GMT 2025
|
PRIMARY | |||
|
LR4LA8YD5Z
Created by
admin on Tue Apr 01 18:56:38 GMT 2025 , Edited by admin on Tue Apr 01 18:56:38 GMT 2025
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
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|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
BRD2(BD2) DOMAIN
Kd
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INHIBITOR -> TARGET | |||
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|
INHIBITOR -> TARGET |
Kd
|
||
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|
INHIBITOR -> TARGET |
A >250x differential binding preference for BDII over BDI
BINDING
|
||
|
INHIBITOR -> TARGET |
IC50
|
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_6] | THREONINE PHOSPHATE | 3L4WX7B1EI | |||
| AMINO ACID SUBSTITUTION | [1_1] | N-ACETYLMETHIONINE | 9J12WX5B6A | |||
| AMINO ACID SUBSTITUTION | [1_37] [1_298] [1_301] [1_305] [1_633] | DEXFOSFOSERINE | VI4F0K069V |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|