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Details

Stereochemistry ABSOLUTE
Molecular Formula C33H43N3O4.2C4H4O4
Molecular Weight 777.8565
Optical Activity UNSPECIFIED
Defined Stereocenters 3 / 3
E/Z Centers 2
Charge 0

SHOW SMILES / InChI
Structure of ACT-280778 maleate

SMILES

OC(=O)\C=C/C(O)=O.OC(=O)\C=C/C(O)=O.COC1=CC=C(OC)C2=C1NC(CCCN(C)CC[C@@]3(C[C@H]4CC[C@@H]3C=C4C5=CC=CC=C5)OC(=O)C(C)C)=N2

InChI

InChIKey=XCOMDWDKJAXYDF-YCAFZAMQSA-N
InChI=1S/C33H43N3O4.2C4H4O4/c1-22(2)32(37)40-33(21-24-13-14-25(33)20-26(24)23-10-7-6-8-11-23)17-19-36(3)18-9-12-29-34-30-27(38-4)15-16-28(39-5)31(30)35-29;2*5-3(6)1-2-4(7)8/h6-8,10-11,15-16,20,22,24-25H,9,12-14,17-19,21H2,1-5H3,(H,34,35);2*1-2H,(H,5,6)(H,7,8)/b;2*2-1-/t24-,25-,33+;;/m1../s1

HIDE SMILES / InChI

Molecular Formula C33H43N3O4
Molecular Weight 545.7122
Charge 0
Count
Stereochemistry ABSOLUTE
Additional Stereochemistry No
Defined Stereocenters 3 / 3
E/Z Centers 0
Optical Activity ( - )

Molecular Formula C4H4O4
Molecular Weight 116.0722
Charge 0
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 1
Optical Activity NONE

Approval Year

Substance Class Chemical
Created
by admin
on Wed Apr 02 20:00:58 GMT 2025
Edited
by admin
on Wed Apr 02 20:00:58 GMT 2025
Record UNII
N2ZP3P57AR
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
ACT-280778B
Preferred Name English
ACT-280778 maleate
Code English
Propanoic acid, 2-methyl-, (1R,2R,4R)-2-[2-[[3-(4,7-dimethoxy-1H-benzimidazol-2-yl)propyl]methylamino]ethyl]-5-phenylbicyclo[2.2.2]oct-5-en-2-yl ester, (2Z)-2-butenedioate (1:2)
Systematic Name English
Code System Code Type Description
PUBCHEM
154701411
Created by admin on Wed Apr 02 20:00:58 GMT 2025 , Edited by admin on Wed Apr 02 20:00:58 GMT 2025
PRIMARY
FDA UNII
N2ZP3P57AR
Created by admin on Wed Apr 02 20:00:58 GMT 2025 , Edited by admin on Wed Apr 02 20:00:58 GMT 2025
PRIMARY
CAS
1537197-53-7
Created by admin on Wed Apr 02 20:00:58 GMT 2025 , Edited by admin on Wed Apr 02 20:00:58 GMT 2025
PRIMARY
SMS_ID
300000047883
Created by admin on Wed Apr 02 20:00:58 GMT 2025 , Edited by admin on Wed Apr 02 20:00:58 GMT 2025
PRIMARY
Related Record Type Details
PARENT -> SALT/SOLVATE
Related Record Type Details
ACTIVE MOIETY