U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 17:29:58 GMT 2025
Edited
by admin
on Tue Apr 01 17:29:58 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
OD27Q24FJ4
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
ARK-1
Preferred Name English
AURORA KINASE A
Common Name English
SERINE/THREONINE-PROTEIN KINASE 15
Common Name English
AURKA
Common Name English
SERINE/THREONINE-PROTEIN KINASE AURORA-A
Common Name English
AURORA 2
Common Name English
AURORA/IPL1-RELATED KINASE 1
Common Name English
SERINE/THREONINE-PROTEIN KINASE 6
Common Name English
AURORA-RELATED KINASE 1
Common Name English
Code System Code Type Description
PHAROS
O14965
Created by admin on Tue Apr 01 17:29:58 GMT 2025 , Edited by admin on Tue Apr 01 17:29:58 GMT 2025
PRIMARY
FDA UNII
OD27Q24FJ4
Created by admin on Tue Apr 01 17:29:58 GMT 2025 , Edited by admin on Tue Apr 01 17:29:58 GMT 2025
PRIMARY
UNIPROT
O14965
Created by admin on Tue Apr 01 17:29:58 GMT 2025 , Edited by admin on Tue Apr 01 17:29:58 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR->OFF-TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
COMPETITIVE INHIBITOR
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
COMPETITIVE INHIBITOR
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_287] [1_288] THREONINE PHOSPHATE 3L4WX7B1EI
AMINO ACID SUBSTITUTION [1_41] [1_51] DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_342] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL