Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 18:23:38 GMT 2025
by
admin
on
Tue Apr 01 18:23:38 GMT 2025
|
| Protein Type | RECEPTOR |
| Protein Sub Type | |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
QV1Q1KK8LA
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Preferred Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
QV1Q1KK8LA
Created by
admin on Tue Apr 01 18:23:38 GMT 2025 , Edited by admin on Tue Apr 01 18:23:38 GMT 2025
|
PRIMARY | |||
|
P41968
Created by
admin on Tue Apr 01 18:23:38 GMT 2025 , Edited by admin on Tue Apr 01 18:23:38 GMT 2025
|
PRIMARY |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_2 |
| N | 1_16 |
| N | 1_28 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
INHIBITOR -> TARGET |
BINDING
Ki
|
||
|
AGONIST -> TARGET |
Ki
|
||
|
AGONIST -> TARGET |
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||
|
AGONIST -> TARGET |
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||
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|
NON-AGONIST->OFF-TARGET |
EC50
|
||
|
|
INHIBITOR -> TARGET |
Ability to block ?-MSH-induced
cAMP production in a CHO cell line expressing hMC3R.
BIOASSAY (CELLULAR)
Ki
|
||
|
AGONIST -> TARGET |
Biased agonist: AP1189 reduced cytokine release but no melanogenesis was induced.
|
||
|
|
AGONIST -> TARGET |
|
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| Molecular Formula | CHEMICAL |
|
||||
| MOL_WEIGHT | CHEMICAL |
|