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Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 15:20:45 GMT 2025
Edited
by admin
on Wed Apr 02 15:20:45 GMT 2025
Protein Type ION CHANNEL
Protein Sub Type GABA RECEPTOR
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
RU3465V8V1
Record Status FAILED
Record Version
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Name Type Language
GABAA RECEPTOR
Common Name English
.GAMMA.-AMINOBUTYRIC ACID A RECEPTOR
Preferred Name English
GABAAR
Common Name English
GAMMA-AMINOBUTYRIC ACID A RECEPTOR
Common Name English
GABA A RECEPTOR
Common Name English
Code System Code Type Description
FDA UNII
RU3465V8V1
Created by admin on Wed Apr 02 15:20:45 GMT 2025 , Edited by admin on Wed Apr 02 15:20:45 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
OFF-TARGET ACTIVITY: INHIBITING LIGAND BINDING TO THE AGBAA CHLORIDE ION CHANNEL
INHIBITOR -> TARGET
OFF-TARGET ACTIVITY: INHIBITING LIGAND BINDING TO GABAA CHLORIDE ION CHANNEL
AGONIST -> TARGET
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AGONIST -> TARGET
SL651498 is a subtype-selective GABAA agonist, which acts as a full agonist at ?2 and ?3 subtypes, and as a partial agonist at ?1 and ?5 (although its action at ?5 subtypes is much weaker than at the others).
POSITIVE ALLOSTERIC MODULATOR (PAM)->TARGET
AGONIST -> TARGET
POSITIVE ALLOSTERIC MODULATOR (PAM)->TARGET
INHIBITOR->OFF-TARGET
OFF-TARGET ACTIVITY: INHIBITING LIGAND BINDING TO THE GABAA CHLORIDE ION CHANNEL
AGONIST -> TARGET
INHIBITOR -> TARGET
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MODULATOR->TARGET
ALLOSTERIC ACTIVATOR
PARTIAL AGONIST->TARGET
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PARTIAL AGONIST->TARGET
INVERSE AGONIST->TARGET
MODULATOR->TARGET
ACTIVATOR -> TARGET
ALLOSTERIC ACTIVATOR
AGONIST -> TARGET
INHIBITOR -> TARGET
AGONIST -> TARGET
MODULATOR->TARGET
INVERSE AGONIST->TARGET
Non selective GABAA inverse agonist. Therapeutic potential is limited by severe side effects (anxiogenic, convulsant, and proconvulsant).
ALLOSTERIC
NEGATIVE ALLOSTERIC MODULATOR (NAM)->TARGET
POSITIVE ALLOSTERIC MODULATOR (PAM)->TARGET
AGONIST -> TARGET
POSITIVE ALLOSTERIC MODULATOR (PAM)->TARGET
ACTIVATOR -> TARGET
MODULATOR
ALLOSTERIC
PARTIAL AGONIST->TARGET
AGONIST -> TARGET
MODULATOR->TARGET
PARTIAL AGONIST->TARGET
PARTIAL AGONIST->TARGET
AGONIST -> TARGET
Positive allosteric modulator on GABAA receptors and, at high concentrations, as a direct agonist of the GABAA receptor.
POSITIVE ALLOSTERIC MODULATOR (PAM)->TARGET
POSITIVE ALLOSTERIC MODULATOR (PAM)->TARGET
POSITIVE ALLOSTERIC MODULATOR (PAM)->TARGET
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL
Molecular Formula CHEMICAL