U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 23:50:14 GMT 2025
Edited
by admin
on Tue Apr 01 23:50:14 GMT 2025
Protein Type ENZYME
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
UR5J2T2G7T
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
FARNESYL TRANSFERASE
Preferred Name English
FARNESYLTRANSFERASE
Common Name English
Code System Code Type Description
UNIPROT
P49356
Created by admin on Tue Apr 01 23:50:14 GMT 2025 , Edited by admin on Tue Apr 01 23:50:14 GMT 2025
MAJOR COMPONENT STRUCTURE/SEQUENCE
FDA UNII
UR5J2T2G7T
Created by admin on Tue Apr 01 23:50:14 GMT 2025 , Edited by admin on Tue Apr 01 23:50:14 GMT 2025
PRIMARY
UNIPROT
P49354
Created by admin on Tue Apr 01 23:50:14 GMT 2025 , Edited by admin on Tue Apr 01 23:50:14 GMT 2025
MAJOR COMPONENT STRUCTURE/SEQUENCE
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
SUBSTRATE -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO_ACID_SUBSTITUTION [2_1] N-TERMINUS N-ACETYLALANINE 26C4VY6Z0M
METAL_BINDING [1_297] [1_299] [1_362] SITE_SPECIFIC ZINC CATION 13S1S8SF37
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL
Molecular Formula CHEMICAL