U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 19:43:39 GMT 2025
Edited
by admin
on Tue Apr 01 19:43:39 GMT 2025
Protein Type KINASE
Protein Sub Type TYROSINE KINASE
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
V094BEF0W8
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
NON-RECEPTOR TYROSINE-PROTEIN KINASE TYK2
Common Name English
TYK2
Preferred Name English
Code System Code Type Description
SMS_ID
100000177932
Created by admin on Tue Apr 01 19:43:39 GMT 2025 , Edited by admin on Tue Apr 01 19:43:39 GMT 2025
PRIMARY
PHAROS
P29597
Created by admin on Tue Apr 01 19:43:39 GMT 2025 , Edited by admin on Tue Apr 01 19:43:39 GMT 2025
PRIMARY
FDA UNII
V094BEF0W8
Created by admin on Tue Apr 01 19:43:39 GMT 2025 , Edited by admin on Tue Apr 01 19:43:39 GMT 2025
PRIMARY
UNIPROT
P29597
Created by admin on Tue Apr 01 19:43:39 GMT 2025 , Edited by admin on Tue Apr 01 19:43:39 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
Tyk2 JH2 ligand
IC50
INHIBITOR -> TARGET
IC50
WEAK INHIBITOR->TARGETF
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
TYK2 JH2 LIGAND
Ki
INHIBITOR -> TARGET
IC50
WEAK INHIBITOR->OFF TARGET
IC50
WEAK INHIBITOR->TARGET
IC50
WEAK INHIBITOR->TARGET
WEAK INHIBITOR->TARGETF
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
WEAK INHIBITOR->TARGETF
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
WEAK INHIBITOR->TARGET
IC50
WEAK INHIBITOR->OFF TARGET
IC50
INHIBITOR -> TARGET
IC50
NON-INHIBITOR->OFF-TARGET
IC50
TARGET -> INHIBITOR
IC50
INHIBITOR -> TARGET
JH1 Binding site
Kd
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IN-VITRO

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_1054] TYROSINE O-PHOSPHATE 2R86C98KDX
AMINO ACID SUBSTITUTION [1_292] [1_604] TYROSINE O-PHOSPHATE 2R86C98KDX
AMINO ACID SUBSTITUTION [1_525] [1_884] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT CHEMICAL