Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 19:43:39 GMT 2025
by
admin
on
Tue Apr 01 19:43:39 GMT 2025
|
| Protein Type | KINASE |
| Protein Sub Type | TYROSINE KINASE |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
V094BEF0W8
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
|
Preferred Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
100000177932
Created by
admin on Tue Apr 01 19:43:39 GMT 2025 , Edited by admin on Tue Apr 01 19:43:39 GMT 2025
|
PRIMARY | |||
|
P29597
Created by
admin on Tue Apr 01 19:43:39 GMT 2025 , Edited by admin on Tue Apr 01 19:43:39 GMT 2025
|
PRIMARY | |||
|
V094BEF0W8
Created by
admin on Tue Apr 01 19:43:39 GMT 2025 , Edited by admin on Tue Apr 01 19:43:39 GMT 2025
|
PRIMARY | |||
|
P29597
Created by
admin on Tue Apr 01 19:43:39 GMT 2025 , Edited by admin on Tue Apr 01 19:43:39 GMT 2025
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
Tyk2 JH2 ligand
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
|
WEAK INHIBITOR->TARGETF |
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
TYK2 JH2 LIGAND
Ki
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
WEAK INHIBITOR->OFF TARGET |
IC50
|
||
|
WEAK INHIBITOR->TARGET |
IC50
|
||
|
WEAK INHIBITOR->TARGET |
|
||
|
WEAK INHIBITOR->TARGETF |
IC50
|
||
|
INHIBITOR -> TARGET |
|
||
|
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
WEAK INHIBITOR->TARGETF |
IC50
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
|
INHIBITOR -> TARGET |
IC50
|
||
|
|
WEAK INHIBITOR->TARGET |
IC50
|
||
|
WEAK INHIBITOR->OFF TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
NON-INHIBITOR->OFF-TARGET |
IC50
|
||
|
|
TARGET -> INHIBITOR |
IC50
|
||
|
INHIBITOR -> TARGET |
JH1 Binding site
Kd
|
||
|
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
IN-VITRO
|
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_1054] | TYROSINE O-PHOSPHATE | 2R86C98KDX | |||
| AMINO ACID SUBSTITUTION | [1_292] [1_604] | TYROSINE O-PHOSPHATE | 2R86C98KDX | |||
| AMINO ACID SUBSTITUTION | [1_525] [1_884] | DEXFOSFOSERINE | VI4F0K069V |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| Molecular Formula | CHEMICAL |
|
||||
| MOL_WEIGHT | CHEMICAL |
|