Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Wed Apr 02 01:22:21 GMT 2025
by
admin
on
Wed Apr 02 01:22:21 GMT 2025
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
VC4EQE3CAI
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
|
Preferred Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
Q00534
Created by
admin on Wed Apr 02 01:22:22 GMT 2025 , Edited by admin on Wed Apr 02 01:22:22 GMT 2025
|
PRIMARY | |||
|
VC4EQE3CAI
Created by
admin on Wed Apr 02 01:22:22 GMT 2025 , Edited by admin on Wed Apr 02 01:22:22 GMT 2025
|
PRIMARY | |||
|
Cyclin-dependent kinase 6
Created by
admin on Wed Apr 02 01:22:22 GMT 2025 , Edited by admin on Wed Apr 02 01:22:22 GMT 2025
|
PRIMARY | |||
|
Q00534
Created by
admin on Wed Apr 02 01:22:22 GMT 2025 , Edited by admin on Wed Apr 02 01:22:22 GMT 2025
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
|
INHIBITOR -> TARGET | |||
|
WEAK INHIBITOR->TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
PRECLINICAL
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
|
||
|
NON-INHIBITOR->OFF TARGET |
IC50
|
||
|
WEAK INHIBITOR->TARGET |
IC50
|
||
|
INHIBITOR -> TARGET | |||
|
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
Ki
|
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|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
CELL-FREE KINASE ASSAY (CDK6/CYCLIN D1)
INHIBITOR
IC50
|
||
|
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INHIBITOR -> TARGET |
|
||
|
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IN-VITRO, IN-VIVO
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_1] | N-ACETYLMETHIONINE | 9J12WX5B6A |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|