Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 23:27:29 GMT 2025
by
admin
on
Tue Apr 01 23:27:29 GMT 2025
|
| Protein Type | REGULATOR PROTEIN |
| Protein Sub Type | |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
W8U7X588F2
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Preferred Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
W8U7X588F2
Created by
admin on Tue Apr 01 23:27:29 GMT 2025 , Edited by admin on Tue Apr 01 23:27:29 GMT 2025
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
INHIBITS MENIN BINDING TO MLL1.
IC50
|
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|
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO_ACID_SUBSTITUTION | [1_599] | SITE_SPECIFIC | THREONINE PHOSPHATE | 3L4WX7B1EI | ||
| AMINO_ACID_SUBSTITUTION | [1_492] [1_548] | SITE_SPECIFIC | DEXFOSFOSERINE | VI4F0K069V |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| Molecular Formula | CHEMICAL |
|
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| MOL_WEIGHT:NUMBER(CALCULATED) | CHEMICAL |
|