U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 23:27:29 GMT 2025
Edited
by admin
on Tue Apr 01 23:27:29 GMT 2025
Protein Type REGULATOR PROTEIN
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
W8U7X588F2
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
MEN1 PROTEIN
Preferred Name English
MENIN
Common Name English
SCG2 PROTEIN
Common Name English
Code System Code Type Description
FDA UNII
W8U7X588F2
Created by admin on Tue Apr 01 23:27:29 GMT 2025 , Edited by admin on Tue Apr 01 23:27:29 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITS MENIN BINDING TO MLL1.
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO_ACID_SUBSTITUTION [1_599] SITE_SPECIFIC THREONINE PHOSPHATE 3L4WX7B1EI
AMINO_ACID_SUBSTITUTION [1_492] [1_548] SITE_SPECIFIC DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL