U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Structurally Diverse
Created
by admin
on Tue Apr 01 21:32:42 GMT 2025
Edited
by admin
on Tue Apr 01 21:32:42 GMT 2025
Source Materials Class ORGANISM
Source Materials Type VIRUS
Source Materials Parent
Part integrase
Fraction Material Type protein
Record UNII
YY6481J2FF
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
HIV-1 INTEGRASE
Preferred Name English
HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 INTEGRASE
Common Name English
Code System Code Type Description
FDA UNII
YY6481J2FF
Created by admin on Tue Apr 01 21:32:42 GMT 2025 , Edited by admin on Tue Apr 01 21:32:42 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
Strand transfer
IC50
INHIBITOR -> TARGET
Mutations (G118R and E138K) confer resistance to MK-2048
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET