Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 16:52:16 GMT 2025
by
admin
on
Tue Apr 01 16:52:16 GMT 2025
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
ZI18M2JAY5
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Preferred Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
ZI18M2JAY5
Created by
admin on Tue Apr 01 16:52:16 GMT 2025 , Edited by admin on Tue Apr 01 16:52:16 GMT 2025
|
PRIMARY | |||
|
P28221
Created by
admin on Tue Apr 01 16:52:16 GMT 2025 , Edited by admin on Tue Apr 01 16:52:16 GMT 2025
|
PRIMARY | |||
|
P28221
Created by
admin on Tue Apr 01 16:52:16 GMT 2025 , Edited by admin on Tue Apr 01 16:52:16 GMT 2025
|
PRIMARY |
| From | To |
|---|---|
| 1_111 | 1_188 |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_5 |
| N | 1_17 |
| N | 1_21 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
LIGAND->TARGET |
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|
INHIBITOR -> TARGET |
ANTAGONIST
|
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AGONIST -> TARGET |
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AGONIST -> TARGET |
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AGONIST -> TARGET |
IC50
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|
AGONIST -> TARGET |
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|
AGONIST -> TARGET |
pKi
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AGONIST -> TARGET |
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|
AGONIST -> TARGET |
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RADIOLIGAND->TARGET |
Ki
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|
AGONIST -> TARGET |
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INHIBITOR -> TARGET |
INHIBITOR
Ki
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||
|
AGONIST -> TARGET |
EC50
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||
|
|
AGONIST -> TARGET |
Natural agonist
Ki
|
||
|
AGONIST -> TARGET |
Eletriptan binds with high affinity to 5-HT1B, 5-HT1D and 5-HT1F receptors, has modest affinity for 5-HT1A, 5-HT1E, 5-HT2B and 5-HT7 receptors
BINDING
|
||
|
INHIBITOR -> TARGET |
INHIBITOR
Ki
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|
AGONIST -> TARGET |
Ki
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|
AGONIST -> TARGET |
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|
AGONIST -> TARGET | |||
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AGONIST -> TARGET |
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|
AGONIST -> TARGET | |||
|
AGONIST -> TARGET | |||
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|
AGONIST -> TARGET |
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| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|
||||
| Molecular Formula | CHEMICAL |
|