Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 19:13:55 GMT 2025
by
admin
on
Tue Apr 01 19:13:55 GMT 2025
|
| Protein Type | KINASE |
| Protein Sub Type | TYROSINE KINASE |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
08S4A2S6FT
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
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Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
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P23458
Created by
admin on Tue Apr 01 19:13:55 GMT 2025 , Edited by admin on Tue Apr 01 19:13:55 GMT 2025
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PRIMARY | |||
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08S4A2S6FT
Created by
admin on Tue Apr 01 19:13:55 GMT 2025 , Edited by admin on Tue Apr 01 19:13:55 GMT 2025
|
PRIMARY | |||
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EC 2.7.10.2
Created by
admin on Tue Apr 01 19:13:55 GMT 2025 , Edited by admin on Tue Apr 01 19:13:55 GMT 2025
|
PRIMARY | |||
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JANUS KINASE 1
Created by
admin on Tue Apr 01 19:13:55 GMT 2025 , Edited by admin on Tue Apr 01 19:13:55 GMT 2025
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
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INHIBITOR -> TARGET |
EC50
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
Calculated IC50 (nM) at 1 mM ATP
COMPETITIVE INHIBITOR
IC50
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
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INHIBITOR->OFF-TARGET |
IC50
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INHIBITOR -> TARGET |
IC50
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INHIBITOR->OFF-TARGET |
Kd
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
ATP at the apparent Km.
IC50
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INHIBITOR -> TARGET |
Potent and selective Janus Kinase 1 Inhibitor, an inhaled treatment for respiratory disease.
IC50
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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NON-INHIBITOR->OFF TARGET |
IC50
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INHIBITOR -> TARGET |
IC50
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INHIBITOR->OFF-TARGET |
IC50
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
IN-VITRO
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
COMPETITIVE INHIBITOR
IC50
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
IC50
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| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| Molecular Formula | CHEMICAL |
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| MOL_WEIGHT:NUMBER AVERAGE(CALCULATED) | CHEMICAL |
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