U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 23:38:34 GMT 2025
Edited
by admin
on Tue Apr 01 23:38:34 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
4M56WLI1MN
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
ANAPLASTIC LYMPHOMA KINASE
Common Name English
CD-246
Preferred Name English
ALK TYROSINE KINASE RECEPTOR
Systematic Name English
ALK
Common Name English
CD246
Code English
Code System Code Type Description
FDA UNII
4M56WLI1MN
Created by admin on Tue Apr 01 23:38:34 GMT 2025 , Edited by admin on Tue Apr 01 23:38:34 GMT 2025
PRIMARY
WIKIPEDIA
ANAPLASTIC LYMPHOMA KINASE
Created by admin on Tue Apr 01 23:38:34 GMT 2025 , Edited by admin on Tue Apr 01 23:38:34 GMT 2025
PRIMARY
UNIPROT
Q9UM73
Created by admin on Tue Apr 01 23:38:34 GMT 2025 , Edited by admin on Tue Apr 01 23:38:34 GMT 2025
PRIMARY
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_151
N 1_226
N 1_267
N 1_306
N 1_393
N 1_406
N 1_427
N 1_545
N 1_553
N 1_609
N 1_691
N 1_790
N 1_845
N 1_846
N 1_868
N 1_968
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR
IC50
INHIBITOR -> TARGET
INHIBITOR
IC50
INHIBITOR -> TARGET
INHIBITOR
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IN-VITRO, IN-VIVO
INHIBITOR -> TARGET
INHIBITOR
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR
IC50
INHIBITOR -> TARGET
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_1060] [1_1074] [1_1078] [1_1113] [1_1260] [1_1489] [1_1586] TYROSINE O-PHOSPHATE 2R86C98KDX
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL