Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 16:59:35 GMT 2025
by
admin
on
Tue Apr 01 16:59:35 GMT 2025
|
| Protein Sub Type | |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
5NJ22TAB5Y
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Preferred Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
P11309
Created by
admin on Tue Apr 01 16:59:35 GMT 2025 , Edited by admin on Tue Apr 01 16:59:35 GMT 2025
|
PRIMARY | |||
|
5NJ22TAB5Y
Created by
admin on Tue Apr 01 16:59:35 GMT 2025 , Edited by admin on Tue Apr 01 16:59:35 GMT 2025
|
PRIMARY | |||
|
87673
Created by
admin on Tue Apr 01 16:59:35 GMT 2025 , Edited by admin on Tue Apr 01 16:59:35 GMT 2025
|
PRIMARY | |||
|
P11309
Created by
admin on Tue Apr 01 16:59:35 GMT 2025 , Edited by admin on Tue Apr 01 16:59:35 GMT 2025
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
Ki
|
||
|
INHIBITOR -> TARGET |
COMPETITIVE INHIBITOR
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
COMPETITIVE INHIBITOR
Ki
|
||
|
|
INHIBITOR -> TARGET |
Kd
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
|
INHIBITOR -> TARGET |
PAN-PIM INHIBITOR
IC50
|
||
|
|
INHIBITOR -> TARGET |
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_99] [1_189] [1_352] | DEXFOSFOSERINE | VI4F0K069V | |||
| AMINO ACID SUBSTITUTION | [1_114] | THREONINE PHOSPHATE | 3L4WX7B1EI |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|