Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 17:59:35 GMT 2025
by
admin
on
Tue Apr 01 17:59:35 GMT 2025
|
| Protein Type | RECEPTOR |
| Protein Sub Type | |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
7H1P16DG5J
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Preferred Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
7H1P16DG5J
Created by
admin on Tue Apr 01 17:59:35 GMT 2025 , Edited by admin on Tue Apr 01 17:59:35 GMT 2025
|
PRIMARY | |||
|
Q13639
Created by
admin on Tue Apr 01 17:59:35 GMT 2025 , Edited by admin on Tue Apr 01 17:59:35 GMT 2025
|
PRIMARY |
| From | To |
|---|---|
| 1_93 | 1_184 |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_7 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
PARTIAL AGONIST->TARGET |
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INHIBITOR -> TARGET |
Kb listed
Kd
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INHIBITOR -> TARGET |
Ki
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AGONIST -> TARGET |
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AGONIST -> TARGET |
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AGONIST -> TARGET |
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INHIBITOR -> TARGET |
INHIBITOR
Ki
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INHIBITOR -> TARGET |
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AGONIST -> TARGET |
Interaction with the 5-HT4 receptor leads to the elevation of cyclic adenosine monophosphate (cAMP) levels in HEK293 cells
EC50
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NON-INHIBITOR -> TRANSPORTER |
Ki
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AGONIST -> TARGET |
BINDING
Ki
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RADIOLIGAND->TARGET |
Kd
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PARTIAL AGONIST->TARGET |
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AGONIST -> TARGET |
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WEAK INHIBITOR->TARGET |
INHIBITOR
Ki
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RADIOLIGAND->TARGET |
Kd
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INHIBITOR -> TARGET |
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AGONIST -> TARGET |
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AGONIST -> TARGET |
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AGONIST -> TARGET |
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AGONIST -> TARGET |
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AGONIST -> TARGET |
BINDING
Ki
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AGONIST -> TARGET |
PARTIAL AGONIST
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AGONIST -> TARGET |
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PARTIAL AGONIST->TARGET |
Has about 50% of the activity of serotonin
Ki
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RADIOLIGAND->TARGET |
IMAGING AGENT
Ki
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AGONIST -> TARGET |
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| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|
||||
| Molecular Formula | CHEMICAL |
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