U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 17:38:05 GMT 2025
Edited
by admin
on Tue Apr 01 17:38:05 GMT 2025
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
7ISX4QDW6N
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
KIAA0043
Preferred Name English
BROMODOMAIN-CONTAINING PROTEIN 3
Common Name English
RING3L
Common Name English
RING3-LIKE PROTEIN
Common Name English
BRD3
Common Name English
Code System Code Type Description
FDA UNII
7ISX4QDW6N
Created by admin on Tue Apr 01 17:38:05 GMT 2025 , Edited by admin on Tue Apr 01 17:38:05 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
Kd
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
A >250x differential binding preference for BDII over BDI
BINDING
INHIBITOR -> TARGET
BRD3(BD2) DOMAIN
Kd

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_262] [1_280] [1_562] DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_1] N-ACETYLSERINE W98518XGZ3
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL