Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 17:43:02 GMT 2025
by
admin
on
Tue Apr 01 17:43:02 GMT 2025
|
| Protein Type | RECEPTOR |
| Protein Sub Type | TYROSINE PROTEIN KINASE |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
8FO9RM2OXK
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
|
Preferred Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
8FO9RM2OXK
Created by
admin on Tue Apr 01 17:43:02 GMT 2025 , Edited by admin on Tue Apr 01 17:43:02 GMT 2025
|
PRIMARY | |||
|
P35916
Created by
admin on Tue Apr 01 17:43:02 GMT 2025 , Edited by admin on Tue Apr 01 17:43:02 GMT 2025
|
PRIMARY |
| From | To |
|---|---|
| 1_27 | 1_87 |
| 1_134 | 1_182 |
| 1_228 | 1_286 |
| 1_421 | 1_510 |
| 1_554 | 1_629 |
| 1_675 | 1_727 |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_9 |
| N | 1_80 |
| N | 1_142 |
| N | 1_227 |
| N | 1_275 |
| N | 1_387 |
| N | 1_491 |
| N | 1_503 |
| N | 1_570 |
| N | 1_659 |
| N | 1_666 |
| N | 1_734 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
|
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|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
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|
INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_1044] [1_1206] [1_1207] [1_1241] [1_1339] | TYROSINE O-PHOSPHATE | 2R86C98KDX | |||
| AMINO ACID SUBSTITUTION | [1_1039] [1_1309] [1_1313] | TYROSINE O-PHOSPHATE | 2R86C98KDX | |||
| AMINO ACID SUBSTITUTION | [1_806] [1_809] [1_829] | TYROSINE O-PHOSPHATE | 2R86C98KDX |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|