U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 17:43:02 GMT 2025
Edited
by admin
on Tue Apr 01 17:43:02 GMT 2025
Protein Type RECEPTOR
Protein Sub Type TYROSINE PROTEIN KINASE
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
8FO9RM2OXK
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR 3
Common Name English
FLT-4
Preferred Name English
FMS-LIKE TYROSINE KINASE 4
Common Name English
TYROSINE-PROTEIN KINASE RECEPTOR FLT4
Common Name English
VEGFR3
Common Name English
Code System Code Type Description
FDA UNII
8FO9RM2OXK
Created by admin on Tue Apr 01 17:43:02 GMT 2025 , Edited by admin on Tue Apr 01 17:43:02 GMT 2025
PRIMARY
UNIPROT
P35916
Created by admin on Tue Apr 01 17:43:02 GMT 2025 , Edited by admin on Tue Apr 01 17:43:02 GMT 2025
PRIMARY
From To
1_27 1_87
1_134 1_182
1_228 1_286
1_421 1_510
1_554 1_629
1_675 1_727
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_9
N 1_80
N 1_142
N 1_227
N 1_275
N 1_387
N 1_491
N 1_503
N 1_570
N 1_659
N 1_666
N 1_734
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_1044] [1_1206] [1_1207] [1_1241] [1_1339] TYROSINE O-PHOSPHATE 2R86C98KDX
AMINO ACID SUBSTITUTION [1_1039] [1_1309] [1_1313] TYROSINE O-PHOSPHATE 2R86C98KDX
AMINO ACID SUBSTITUTION [1_806] [1_809] [1_829] TYROSINE O-PHOSPHATE 2R86C98KDX
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL