Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 19:04:29 GMT 2025
by
admin
on
Tue Apr 01 19:04:29 GMT 2025
|
| Protein Type | KINASE |
| Protein Sub Type | TYROSINE KINASE |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
9LLR266790
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
|
Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
JANUS KINASE 3
Created by
admin on Tue Apr 01 19:04:29 GMT 2025 , Edited by admin on Tue Apr 01 19:04:29 GMT 2025
|
PRIMARY | |||
|
9LLR266790
Created by
admin on Tue Apr 01 19:04:29 GMT 2025 , Edited by admin on Tue Apr 01 19:04:29 GMT 2025
|
PRIMARY | |||
|
EC 2.7.10.2
Created by
admin on Tue Apr 01 19:04:29 GMT 2025 , Edited by admin on Tue Apr 01 19:04:29 GMT 2025
|
PRIMARY | |||
|
479898-67-4
Created by
admin on Tue Apr 01 19:04:29 GMT 2025 , Edited by admin on Tue Apr 01 19:04:29 GMT 2025
|
PRIMARY | |||
|
480546-04-1
Created by
admin on Tue Apr 01 19:04:29 GMT 2025 , Edited by admin on Tue Apr 01 19:04:29 GMT 2025
|
ALTERNATIVE |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
|
INHIBITOR -> TARGET |
IC50
|
||
|
|
INHIBITOR -> TARGET |
IC50
|
||
|
WEAK INHIBITOR->TARGET |
IC50
|
||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET | |||
|
|
INHIBITOR -> TARGET |
|
||
|
WEAK INHIBITOR->TARGET |
IC50
|
||
|
|
WEAK INHIBITOR->TARGETF |
|
||
|
|
NON-INHIBITOR->OFF-TARGET |
IC50
|
||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
WEAK INHIBITOR->TARGETF |
IC50
|
||
|
WEAK INHIBITOR->TARGETF |
IC50
|
||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
|
OFF TARGET->NON-INHIBITOR |
IC50
|
||
|
|
WEAK INHIBITOR->TARGETF |
IC50
|
||
|
WEAK INHIBITOR->TARGET |
COMPETITIVE INHIBITOR
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET | |||
|
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
|
||
|
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET | |||
|
NON-INHIBITOR->OFF TARGET |
IC50
|
||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR->OFF-TARGET |
Kd
|
||
|
INHIBITOR -> TARGET |
IN-VIVO
|
||
|
INHIBITOR -> TARGET | |||
|
|
WEAK INHIBITOR->TARGET | |||
|
INHIBITOR -> TARGET |
IRREVERSIBLE INHIBITOR
k(inactivation)
|
||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_17] | SERINE | DEXFOSFOSERINE | VI4F0K069V |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT:NUMBER AVERAGE(CALCULATED) | CHEMICAL |
|
||||
| Molecular Formula | CHEMICAL |
|