U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 13:59:46 GMT 2025
Edited
by admin
on Wed Apr 02 13:59:46 GMT 2025
Protein Type COAGULATION FACTOR
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
DQP38C562S
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
Human recombinant factor VIIa variant (P10Q, K32E, T106N, V253N), desialylated
Preferred Name English
CT-001
Common Name English
Classification Tree Code System Code
FDA ORPHAN DRUG 782420
Created by admin on Wed Apr 02 13:59:46 GMT 2025 , Edited by admin on Wed Apr 02 13:59:46 GMT 2025
Code System Code Type Description
FDA UNII
DQP38C562S
Created by admin on Wed Apr 02 13:59:46 GMT 2025 , Edited by admin on Wed Apr 02 13:59:46 GMT 2025
PRIMARY
From To
1_7 1_12
1_26 1_42
1_158 1_177
1_188 1_216
2_17 2_22
2_50 2_61
2_55 2_70
2_72 2_81
2_91 2_102
2_98 2_112
2_114 2_127
1_110 2_135
Glycosylation Type MAMMALIAN, DESIALYLATED
Glycosylation Link Type Site
N 1_170
N 2_145
O 2_52
O 2_60
Related Record Type Details
TARGET -> ACTIVATOR
Related Record Type Details
ACTIVE MOIETY

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO_ACID_SUBSTITUTION [2_63] SITE_SPECIFIC ASP .BETA.-HYDROXY-L-ASPARTIC ACID, ERYTHRO- GDV0MSK2SG
AMINO_ACID_SUBSTITUTION [2_6] [2_7] [2_14] [2_16] [2_19] [2_20] [2_25] [2_26] [2_29] [2_35] SITE_SPECIFIC GLU .GAMMA.-CARBOXYGLUTAMIC ACID 16FQV4RZKL
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL