Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Wed Apr 02 02:07:31 GMT 2025
by
admin
on
Wed Apr 02 02:07:31 GMT 2025
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
F5Q48O042G
|
| Record Status |
Validated (UNII)
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| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
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Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
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F5Q48O042G
Created by
admin on Wed Apr 02 02:07:31 GMT 2025 , Edited by admin on Wed Apr 02 02:07:31 GMT 2025
|
PRIMARY | |||
|
P51681
Created by
admin on Wed Apr 02 02:07:31 GMT 2025 , Edited by admin on Wed Apr 02 02:07:31 GMT 2025
|
PRIMARY |
| From | To |
|---|---|
| 1_101 | 1_178 |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| O | 1_6 |
| O | 1_7 |
| O | 1_16 |
| O | 1_17 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
Did not reported any cardiovascular risk, but it was failed because of unclear reasons in
a phase IIb study for rheumatoid arthritis.
Ki
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
Blocks HIV infection
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Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_336] [1_337] [1_342] [1_349] | DEXFOSFOSERINE | VI4F0K069V | |||
| AMINO ACID SUBSTITUTION | [1_3] [1_10] [1_14] [1_15] | TYROSINE O-SULFATE | 29166358BF |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|