U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 02:07:31 GMT 2025
Edited
by admin
on Wed Apr 02 02:07:31 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
F5Q48O042G
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
CC-CKR-5
Preferred Name English
C-C CHEMOKINE RECEPTOR TYPE 5
Common Name English
CD-195
Common Name English
CD195
Common Name English
CCR-5
Common Name English
CCR5
Common Name English
CHEMR-13
Common Name English
CHEMR13
Common Name English
Code System Code Type Description
FDA UNII
F5Q48O042G
Created by admin on Wed Apr 02 02:07:31 GMT 2025 , Edited by admin on Wed Apr 02 02:07:31 GMT 2025
PRIMARY
UNIPROT
P51681
Created by admin on Wed Apr 02 02:07:31 GMT 2025 , Edited by admin on Wed Apr 02 02:07:31 GMT 2025
PRIMARY
From To
1_101 1_178
Glycosylation Type HUMAN
Glycosylation Link Type Site
O 1_6
O 1_7
O 1_16
O 1_17
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
Did not reported any cardiovascular risk, but it was failed because of unclear reasons in a phase IIb study for rheumatoid arthritis.
Ki
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
Blocks HIV infection

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_336] [1_337] [1_342] [1_349] DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_3] [1_10] [1_14] [1_15] TYROSINE O-SULFATE 29166358BF
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL