AZILSARTAN

U.S. Department of Health & Human Services Divider Arrow

National Institutes of Health Divider Arrow

NCATS

Details

Stereochemistry	ACHIRAL
Molecular Formula	C25H20N4O5
Molecular Weight	456.4501
Optical Activity	NONE
Defined Stereocenters	0 / 0
E/Z Centers	0
Charge	0

SHOW SMILES / InChI

Structure of AZILSARTAN

Structure Search

SMILES

CCOC1=NC2=C(N1CC3=CC=C(C=C3)C4=CC=CC=C4C5=NOC(=O)N5)C(=CC=C2)C(O)=O

InChI

InChIKey=KGSXMPPBFPAXLY-UHFFFAOYSA-N

InChI=1S/C25H20N4O5/c1-2-33-24-26-20-9-5-8-19(23(30)31)21(20)29(24)14-15-10-12-16(13-11-15)17-6-3-4-7-18(17)22-27-25(32)34-28-22/h3-13H,2,14H2,1H3,(H,30,31)(H,27,28,32)

HIDE SMILES / InChI

Molecular Formula	C25H20N4O5
Molecular Weight	456.4501
Charge	0
Count

Stereochemistry	ACHIRAL
Additional Stereochemistry	No
Defined Stereocenters	0 / 0
E/Z Centers	0
Optical Activity	NONE

Approval Year

Substance Class	Chemical Created by `admin` on `Fri Dec 15 15:56:11 UTC 2023` Edited by `admin` on `Fri Dec 15 15:56:11 UTC 2023`
Record UNII	F9NUX55P23
Record Status	`Validated (UNII)`
Record Version

Download

Name

Type

Language

AZILSARTAN

Official Name

English

AZILSARTAN [MART.]

Common Name

English

TAK-536

Code

English

AZILSARTAN [MI]

Common Name

English

azilsartan [INN]

Common Name

English

1H-BENZIMIDAZOLE-7-CARBOXYLIC ACID, 1-((2'-(2,5-DIHYDRO-5-OXO-1,2,4-OXADIAZOL- 3-YL)(1,1'-BIPHENYL)-4-YL)METHYL)-2-ETHOXY-

Common Name

English

AZILSARTAN [JAN]

Common Name

English

2-ETHOXY-1-((2'-(5-OXO-2,5-DIHYDRO-1,2,4-OXADIAZOL-3-YL)BIPHENYL-4-YL)METHYL)-1H-BENZIMIDAZOLE-7-CARBOXYLIC ACID

Systematic Name

English

AZILSARTAN [VANDF]

Common Name

English

Azilsartan [WHO-DD]

Common Name

English

AZILSARTAN [USAN]

Common Name

English

Classification Tree Code System Code

NDF-RT

N0000175561

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

NCI_THESAURUS

C66930

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

LIVERTOX

NBK548036

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

Code System Code Type Description

ChEMBL

CHEMBL57242

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

PRIMARY

MERCK INDEX

m2173

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

PRIMARY

Merck Index

PUBCHEM

135415867

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

PRIMARY

USAN

TT-131

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

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LACTMED

Azilsartan

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

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INN

8724

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

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NDF-RT

N0000178477

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

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Decreased Blood Pressure [PE]

CHEBI

68850

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

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CAS

147403-03-0

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

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EVMPD

SUB31561

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

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EPA CompTox

DTXSID70163712

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

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MESH

C521273

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

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RXCUI

1091643

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

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RxNorm

DAILYMED

F9NUX55P23

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

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FDA UNII

F9NUX55P23

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

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DRUG BANK

DB08822

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

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NDF-RT

N0000180999

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

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Angiotensin 2 Type 1 Receptor Antagonists [MoA]

SMS_ID

100000124198

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

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NCI_THESAURUS

C75107

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

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HSDB

8208

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

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WIKIPEDIA

AZILSARTAN

Created by admin on Fri Dec 15 15:56:11 UTC 2023 , Edited by admin on Fri Dec 15 15:56:11 UTC 2023

PRIMARY

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Amount:

Name	Property Type	Amount	Referenced Substance	Defining	Parameters	References
Volume of Distribution	PHARMACOKINETIC

Tmax	PHARMACOKINETIC

Biological Half-life	PHARMACOKINETIC