U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 17:28:46 GMT 2025
Edited
by admin
on Wed Apr 02 17:28:46 GMT 2025
Protein Type ENZYME
Protein Sub Type
Sequence Type COMPLETE
Record UNII
H6Y3CRX3LC
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
Rinvecalinase Alfa
INN   USAN  
Official Name English
DM-199
Preferred Name English
Tissue kallikrein (recombinant human clone DM199)
Common Name English
RINVECALINASE ALFA [USAN]
Common Name English
rinvecalinase alfa [INN]
Common Name English
DM199
Code English
human kallikrein-1 (tissue kallikrein, KLK1, EC:3.4.21.35) mature form, engineered variant (E 121>Q, A 164>V) produced in Chinese hamster ovary (CHO) cells, glycoform alfa kallikrein-1 analogue
Common Name English
Code System Code Type Description
NCI_THESAURUS
C199219
Created by admin on Wed Apr 02 17:28:46 GMT 2025 , Edited by admin on Wed Apr 02 17:28:46 GMT 2025
PRIMARY
USAN
LM-259
Created by admin on Wed Apr 02 17:28:46 GMT 2025 , Edited by admin on Wed Apr 02 17:28:46 GMT 2025
PRIMARY
SMS_ID
300000051844
Created by admin on Wed Apr 02 17:28:46 GMT 2025 , Edited by admin on Wed Apr 02 17:28:46 GMT 2025
PRIMARY
FDA UNII
H6Y3CRX3LC
Created by admin on Wed Apr 02 17:28:46 GMT 2025 , Edited by admin on Wed Apr 02 17:28:46 GMT 2025
PRIMARY
CAS
2419877-37-3
Created by admin on Wed Apr 02 17:28:46 GMT 2025 , Edited by admin on Wed Apr 02 17:28:46 GMT 2025
PRIMARY
INN
12246
Created by admin on Wed Apr 02 17:28:46 GMT 2025 , Edited by admin on Wed Apr 02 17:28:46 GMT 2025
PRIMARY
From To
1_186 1_211
1_161 1_175
1_129 1_196
1_26 1_42
1_7 1_150
Glycosylation Type MAMMALIAN
Glycosylation Link Type Site
N 1_78
N 1_84
N 1_141
Related Record Type Details
TARGET->ENZYME REPLACEMENT
PARENT -> DERIVATIVE
Related Record Type Details
ACTIVE MOIETY
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL
Molecular Formula CHEMICAL