Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 18:12:24 GMT 2025
by
admin
on
Tue Apr 01 18:12:24 GMT 2025
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
L1Q8TMD5IZ
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
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Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
Q03181
Created by
admin on Tue Apr 01 18:12:24 GMT 2025 , Edited by admin on Tue Apr 01 18:12:24 GMT 2025
|
PRIMARY | |||
|
L1Q8TMD5IZ
Created by
admin on Tue Apr 01 18:12:24 GMT 2025 , Edited by admin on Tue Apr 01 18:12:24 GMT 2025
|
PRIMARY | |||
|
Q03181
Created by
admin on Tue Apr 01 18:12:24 GMT 2025 , Edited by admin on Tue Apr 01 18:12:24 GMT 2025
|
PRIMARY |
| Linkage Type | Residue Index | |||
|---|---|---|---|---|
| COORDINATION COMPOUND | 1_74 | 1_77 | 1_91 | 1_94 |
| COORDINATION COMPOUND | 1_111 | 1_115 | 1_125 | 1_128 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
PARTIAL AGONIST->TARGET |
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AGONIST -> TARGET |
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INHIBITOR -> TARGET |
IRREVERSIBLE INHIBITOR
IC50
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AGONIST -> TARGET | |||
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AGONIST -> TARGET |
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AGONIST -> TARGET |
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INHIBITOR -> TARGET |
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AGONIST -> TARGET |
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AGONIST -> TARGET |
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AGONIST -> TARGET |
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AGONIST -> TARGET | |||
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ACTIVATOR -> TARGET | |||
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AGONIST -> TARGET |
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AGONIST -> TARGET |
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AGONIST -> TARGET |
AGONIST
EC50
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AGONIST -> TARGET |
SELECTIVE
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AGONIST -> TARGET |
SELECTIVE
EC50
|
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO_ACID_SUBSTITUTION | [1_111] [1_115] [1_125] [1_128] | SITE_SPECIFIC | C4-TYPE ZINC FINGER | C56TF4V7OP | ||
| AMINO_ACID_SUBSTITUTION | [1_74] [1_77] [1_91] [1_94] | SITE_SPECIFIC | C4-TYPE ZINC FINGER | C56TF4V7OP |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|