Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 18:35:25 GMT 2025
by
admin
on
Tue Apr 01 18:35:25 GMT 2025
|
| Protein Type | ENZYME |
| Protein Sub Type | |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
LZ0P651QHS
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
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| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
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LZ0P651QHS
Created by
admin on Tue Apr 01 18:35:25 GMT 2025 , Edited by admin on Tue Apr 01 18:35:25 GMT 2025
|
PRIMARY | |||
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Q9UGN5
Created by
admin on Tue Apr 01 18:35:25 GMT 2025 , Edited by admin on Tue Apr 01 18:35:25 GMT 2025
|
PRIMARY | |||
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Q9UGN5
Created by
admin on Tue Apr 01 18:35:25 GMT 2025 , Edited by admin on Tue Apr 01 18:35:25 GMT 2025
|
PRIMARY | |||
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PARP2
Created by
admin on Tue Apr 01 18:35:25 GMT 2025 , Edited by admin on Tue Apr 01 18:35:25 GMT 2025
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
NON-INHIBITOR->OFF TARGET |
Kd
|
||
|
INHIBITOR -> TARGET |
The selective inhibition of MPH against PARPs analyzed by biotinylated NAD+ -based luminescence assays
IC50
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
IC50
|
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NON-INHIBITOR->OFF TARGET |
Kd
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||
|
INHIBITOR -> TARGET |
IC50
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|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| Other | [1_37] [1_38] | SITE_SPECIFIC | N6-ACETYLLYSINE | 470AD5VY1X | ||
| AMINO ACID SUBSTITUTION | [1_226] [1_232] | SITE_SPECIFIC | DEXFOSFOSERINE | VI4F0K069V |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|