U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 18:23:16 GMT 2025
Edited
by admin
on Tue Apr 01 18:23:16 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
SX1JPI95HB
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
ACTIVIN RECEPTOR TYPE-1
Common Name English
ACTIVIN RECEPTOR-LIKE KINASE 2
Preferred Name English
SERINE/THREONINE-PROTEIN KINASE RECEPTOR R1
Systematic Name English
ALK-2
Common Name English
ALK2
Common Name English
SKR-1
Common Name English
SKR1
Common Name English
TSR-I
Common Name English
TGF-B SUPERFAMILY RECEPTOR TYPE I
Common Name English
ACVR1
Common Name English
Code System Code Type Description
FDA UNII
SX1JPI95HB
Created by admin on Tue Apr 01 18:23:16 GMT 2025 , Edited by admin on Tue Apr 01 18:23:16 GMT 2025
PRIMARY
UNIPROT
Q04771
Created by admin on Tue Apr 01 18:23:16 GMT 2025 , Edited by admin on Tue Apr 01 18:23:16 GMT 2025
PRIMARY
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_82
Related Record Type Details
INHIBITOR -> TARGET
AGONIST -> TARGET
Type I receptor ACVR1, type II receptor ACVR2A and BMP-7 agonist proteins must form a complex to initiate the canonical BMP signaling cascade.
INHIBITOR -> TARGET
INHIBITOR -> TARGET
LIGAND->TARGET
AGONIST -> TARGET
Type I receptor ACVR1, type II receptor ACVR2A and BMP-7 agonist proteins must form a complex to initiate the canonical BMP signaling cascade.
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
inhibitor of both mutated ALK2 and wild type (wt)ALK2
INHIBITOR -> TARGET
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_481] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL
Molecular Formula CHEMICAL