Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 16:49:57 GMT 2025
by
admin
on
Tue Apr 01 16:49:57 GMT 2025
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
Y154T023U0
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
|
Preferred Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
Y154T023U0
Created by
admin on Tue Apr 01 16:49:57 GMT 2025 , Edited by admin on Tue Apr 01 16:49:57 GMT 2025
|
PRIMARY | |||
|
P29274
Created by
admin on Tue Apr 01 16:49:57 GMT 2025 , Edited by admin on Tue Apr 01 16:49:57 GMT 2025
|
PRIMARY | |||
|
P29274
Created by
admin on Tue Apr 01 16:49:57 GMT 2025 , Edited by admin on Tue Apr 01 16:49:57 GMT 2025
|
PRIMARY |
| From | To |
|---|---|
| 1_71 | 1_159 |
| 1_74 | 1_146 |
| 1_77 | 1_166 |
| 1_259 | 1_262 |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_154 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
AGONIST -> TARGET |
BINDING
Kd
|
||
|
INHIBITOR -> TARGET | |||
|
AGONIST -> TARGET |
|
||
|
INHIBITOR -> TARGET |
BINDING
IC50
|
||
|
|
AGONIST -> TARGET |
|
||
|
|
INHIBITOR -> TARGET |
IC50
|
||
|
|
INHIBITOR -> TARGET | |||
|
AGONIST -> TARGET |
|
||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
Approximately 1000-fold more selective
over other ARs.
Ki
|
||
|
INHIBITOR -> TARGET |
Ki
|
||
|
INHIBITOR -> TARGET |
Highly selective over hA2B Ki = 1110 nM.
Ki
|
||
|
|
INHIBITOR -> TARGET |
ANTAGONIST
IC50
|
||
|
RADIOLIGAND->TARGET |
|
||
|
INHIBITOR -> TARGET |
ANTAGONIST
Ki
|
||
|
AGONIST -> TARGET |
BINDING
IC50
|
||
|
RADIOLIGAND->TARGET |
BINDING
Kd
|
||
|
|
INHIBITOR -> TARGET |
Ki
|
||
|
|
WEAK AGONIST->OFF TARGET |
Rat brain receptor
BINDING
Ki
|
||
|
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
|
||
|
RADIOLIGAND->TARGET |
Ki
|
||
|
|
INHIBITOR -> TARGET |
BINDING
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
selective antagonsist
Ki
|
||
|
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
BINDING
IC50
|
||
|
INHIBITOR -> TARGET |
Showed high selectivity over other adenosine receptors.
Ki
|
||
|
WEAK INHIBITOR->TARGET |
Nonselective adenosine receptor antagonist. May be responsible for pain relief.
Ki
|
||
|
AGONIST -> TARGET |
|
||
|
INHIBITOR -> TARGET |
Kb actually
Ki
|
||
|
RADIOLIGAND->TARGET |
Kd
|
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|
AGONIST -> TARGET |
|
||
|
INVERSE AGONIST->TARGET |
EC50
|
||
|
INHIBITOR -> TARGET |
|
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|
INHIBITOR -> TARGET |
IC50
|
||
|
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
ANTAGONIST
Ki
|
||
|
AGONIST -> TARGET |
|
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| Molecular Formula | CHEMICAL |
|
||||
| MOL_WEIGHT | CHEMICAL |
|