U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 19:19:24 GMT 2025
Edited
by admin
on Tue Apr 01 19:19:24 GMT 2025
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
228L4H44D3
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
MAPK/ERK KINASE KINASE 2
Preferred Name English
MITOGEN-ACTIVATED PROTEIN KINASE KINASE KINASE 2
Common Name English
MEKK 2
Common Name English
MEKK2
Common Name English
MEK KINASE 2
Common Name English
MAPKKK2
Common Name English
Code System Code Type Description
PHAROS
Q9Y2U5
Created by admin on Tue Apr 01 19:19:24 GMT 2025 , Edited by admin on Tue Apr 01 19:19:24 GMT 2025
PRIMARY
FDA UNII
228L4H44D3
Created by admin on Tue Apr 01 19:19:24 GMT 2025 , Edited by admin on Tue Apr 01 19:19:24 GMT 2025
PRIMARY
UNIPROT
Q9Y2U5
Created by admin on Tue Apr 01 19:19:24 GMT 2025 , Edited by admin on Tue Apr 01 19:19:24 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
ALLOSTERIC INHIBITOR
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_26] [1_153] [1_159] [1_164] [1_239] [1_297] [1_331] [1_344] [1_349] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL