U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 23:47:22 GMT 2025
Edited
by admin
on Tue Apr 01 23:47:22 GMT 2025
Protein Type ENZYME
Protein Sub Type DEACETYLASE
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
7YNS2RVD5Q
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
HISTONE DEACETYLASE 3
Common Name English
HDAC3
Preferred Name English
Code System Code Type Description
UNIPROT
O15379
Created by admin on Tue Apr 01 23:47:22 GMT 2025 , Edited by admin on Tue Apr 01 23:47:22 GMT 2025
PRIMARY
FDA UNII
7YNS2RVD5Q
Created by admin on Tue Apr 01 23:47:22 GMT 2025 , Edited by admin on Tue Apr 01 23:47:22 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
WEAK INHIBITOR->TARGET
IC50
INHIBITOR -> TARGET
Pan HDAC inhibitor
INHIBITOR -> TARGET
IC50
WEAK INHIBITOR->TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IN-VIVO
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_424] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL
Molecular Formula CHEMICAL