U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 16:36:37 GMT 2025
Edited
by admin
on Tue Apr 01 16:36:37 GMT 2025
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
S344CKA15F
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
FIBROBLAST GROWTH FACTOR RECEPTOR 2
Common Name English
FGFR-2
Preferred Name English
FGFR2
Common Name English
KERATINOCYTE GROWTH FACTOR RECEPTOR
Common Name English
Code System Code Type Description
PHAROS
P21802
Created by admin on Tue Apr 01 16:36:37 GMT 2025 , Edited by admin on Tue Apr 01 16:36:37 GMT 2025
PRIMARY
FDA UNII
S344CKA15F
Created by admin on Tue Apr 01 16:36:37 GMT 2025 , Edited by admin on Tue Apr 01 16:36:37 GMT 2025
PRIMARY
UNIPROT
P21802
Created by admin on Tue Apr 01 16:36:37 GMT 2025 , Edited by admin on Tue Apr 01 16:36:37 GMT 2025
PRIMARY
From To
1_41 1_86
1_158 1_210
1_257 1_321
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_62
N 1_102
N 1_207
N 1_220
N 1_244
N 1_276
N 1_297
N 1_310
Related Record Type Details
INHIBITOR -> TARGET
MUTANT->PARENT
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
at higher concentrations that were still clinically achievable
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
CONJUGATED TOXIN->TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_445] [1_565] [1_567] [1_635] [1_636] [1_748] TYROSINE O-PHOSPHATE 2R86C98KDX
AMINO ACID SUBSTITUTION [1_759] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL