Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 16:36:37 GMT 2025
by
admin
on
Tue Apr 01 16:36:37 GMT 2025
|
| Protein Sub Type | |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
S344CKA15F
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
|
Preferred Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
P21802
Created by
admin on Tue Apr 01 16:36:37 GMT 2025 , Edited by admin on Tue Apr 01 16:36:37 GMT 2025
|
PRIMARY | |||
|
S344CKA15F
Created by
admin on Tue Apr 01 16:36:37 GMT 2025 , Edited by admin on Tue Apr 01 16:36:37 GMT 2025
|
PRIMARY | |||
|
P21802
Created by
admin on Tue Apr 01 16:36:37 GMT 2025 , Edited by admin on Tue Apr 01 16:36:37 GMT 2025
|
PRIMARY |
| From | To |
|---|---|
| 1_41 | 1_86 |
| 1_158 | 1_210 |
| 1_257 | 1_321 |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_62 |
| N | 1_102 |
| N | 1_207 |
| N | 1_220 |
| N | 1_244 |
| N | 1_276 |
| N | 1_297 |
| N | 1_310 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
|
INHIBITOR -> TARGET | |||
|
MUTANT->PARENT |
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||
|
INHIBITOR -> TARGET |
IC50
|
||
|
INHIBITOR -> TARGET |
at higher concentrations that were still clinically achievable
|
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|
INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
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||
|
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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CONJUGATED TOXIN->TARGET | |||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_445] [1_565] [1_567] [1_635] [1_636] [1_748] | TYROSINE O-PHOSPHATE | 2R86C98KDX | |||
| AMINO ACID SUBSTITUTION | [1_759] | DEXFOSFOSERINE | VI4F0K069V |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|