U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Mon Mar 31 22:29:07 GMT 2025
Edited
by admin
on Mon Mar 31 22:29:07 GMT 2025
Protein Type MONOCLONAL ANTIBODY
Protein Sub Type IGG1
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
RJW23BQ0KW
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
FPA-144
Preferred Name English
BEMARITUZUMAB
INN  
Official Name English
bemarituzumab [INN]
Common Name English
ANTI-FGFR2 MONOCLONAL ANTIBODY FPA144
Common Name English
Bemarituzumab [WHO-DD]
Common Name English
Classification Tree Code System Code
NCI_THESAURUS C129822
Created by admin on Mon Mar 31 22:29:07 GMT 2025 , Edited by admin on Mon Mar 31 22:29:07 GMT 2025
FDA ORPHAN DRUG 527716
Created by admin on Mon Mar 31 22:29:07 GMT 2025 , Edited by admin on Mon Mar 31 22:29:07 GMT 2025
NCI_THESAURUS C133879
Created by admin on Mon Mar 31 22:29:07 GMT 2025 , Edited by admin on Mon Mar 31 22:29:07 GMT 2025
Code System Code Type Description
FDA UNII
RJW23BQ0KW
Created by admin on Mon Mar 31 22:29:07 GMT 2025 , Edited by admin on Mon Mar 31 22:29:07 GMT 2025
PRIMARY
SMS_ID
100000181859
Created by admin on Mon Mar 31 22:29:07 GMT 2025 , Edited by admin on Mon Mar 31 22:29:07 GMT 2025
PRIMARY
NCI_THESAURUS
C120040
Created by admin on Mon Mar 31 22:29:07 GMT 2025 , Edited by admin on Mon Mar 31 22:29:07 GMT 2025
PRIMARY
INN
10681
Created by admin on Mon Mar 31 22:29:07 GMT 2025 , Edited by admin on Mon Mar 31 22:29:07 GMT 2025
PRIMARY
CAS
1952272-74-0
Created by admin on Mon Mar 31 22:29:07 GMT 2025 , Edited by admin on Mon Mar 31 22:29:07 GMT 2025
PRIMARY
From To
1_22 1_96
1_141 1_197
1_258 1_318
1_364 1_422
2_22 2_96
2_141 2_197
2_258 2_318
2_364 2_422
1_217 3_214
2_217 4_214
1_223 2_223
1_226 2_226
3_23 3_88
3_134 3_194
4_23 4_88
4_134 4_194
Glycosylation Type MAMMALIAN, AFUCOSYLATED
Glycosylation Link Type Site
N 1_294
N 2_294
Related Record Type Details
TARGET -> INHIBITOR
Related Record Type Details
ACTIVE MOIETY

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO_ACID_SUBSTITUTION [1_1] N-TERMINUS PIDOLIC ACID SZB83O1W42
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL
Molecular Formula CHEMICAL