U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 17:33:15 GMT 2025
Edited
by admin
on Tue Apr 01 17:33:15 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
1788PW098Q
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
FRAP
Preferred Name English
SERINE/THREONINE-PROTEIN KINASE MTOR
Common Name English
MTOR
Common Name English
RAFT1
Common Name English
FRAP2
Common Name English
MAMMALIAN TARGET OF RAPAMYCIN
Common Name English
RAPAMYCIN AND FKBP12 TARGET 1
Common Name English
FKBP12-RAPAMYCIN COMPLEX-ASSOCIATED PROTEIN
Common Name English
FK506-BINDING PROTEIN 12-RAPAMYCIN COMPLEX-ASSOCIATED PROTEIN 1
Common Name English
Code System Code Type Description
SMS_ID
100000178389
Created by admin on Tue Apr 01 17:33:15 GMT 2025 , Edited by admin on Tue Apr 01 17:33:15 GMT 2025
PRIMARY
UNIPROT
P42345
Created by admin on Tue Apr 01 17:33:15 GMT 2025 , Edited by admin on Tue Apr 01 17:33:15 GMT 2025
PRIMARY
FDA UNII
1788PW098Q
Created by admin on Tue Apr 01 17:33:15 GMT 2025 , Edited by admin on Tue Apr 01 17:33:15 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
ALLOSTERIC INHIBITOR
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
clinically relevant ATP site inhibitor of mTOR
COMPETITIVE INHIBITOR
Ki
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
Using native mTOR enzyme complexes extracted from HeLa cells
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL