Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 17:33:15 GMT 2025
by
admin
on
Tue Apr 01 17:33:15 GMT 2025
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
1788PW098Q
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
100000178389
Created by
admin on Tue Apr 01 17:33:15 GMT 2025 , Edited by admin on Tue Apr 01 17:33:15 GMT 2025
|
PRIMARY | |||
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P42345
Created by
admin on Tue Apr 01 17:33:15 GMT 2025 , Edited by admin on Tue Apr 01 17:33:15 GMT 2025
|
PRIMARY | |||
|
1788PW098Q
Created by
admin on Tue Apr 01 17:33:15 GMT 2025 , Edited by admin on Tue Apr 01 17:33:15 GMT 2025
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
ALLOSTERIC INHIBITOR
|
||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
|
||
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INHIBITOR -> TARGET |
IC50
|
||
|
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
clinically relevant ATP site inhibitor of mTOR
COMPETITIVE INHIBITOR
Ki
|
||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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||
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INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
Using native mTOR
enzyme complexes extracted from HeLa cells
IC50
|
||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
|
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| Molecular Formula | CHEMICAL |
|
||||
| MOL_WEIGHT:NUMBER(CALCULATED) | CHEMICAL |
|