Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 16:49:13 GMT 2025
by
admin
on
Tue Apr 01 16:49:13 GMT 2025
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
2VXO9I489U
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
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Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
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2VXO9I489U
Created by
admin on Tue Apr 01 16:49:13 GMT 2025 , Edited by admin on Tue Apr 01 16:49:13 GMT 2025
|
PRIMARY | |||
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P07333
Created by
admin on Tue Apr 01 16:49:13 GMT 2025 , Edited by admin on Tue Apr 01 16:49:13 GMT 2025
|
PRIMARY |
| From | To |
|---|---|
| 1_23 | 1_65 |
| 1_108 | 1_158 |
| 1_205 | 1_259 |
| 1_400 | 1_466 |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_26 |
| N | 1_54 |
| N | 1_134 |
| N | 1_221 |
| N | 1_256 |
| N | 1_283 |
| N | 1_316 |
| N | 1_334 |
| N | 1_393 |
| N | 1_409 |
| N | 1_461 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
Selective exhibited nanomolar potency for
inhibition of CSF-1R but not other 453 kinases
tested.
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
Prevents the binding of both colony stimulating factor 1 (CSF-1) and interleukin 34 (IL-34) to CSF-1R
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET | |||
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TARGET -> INHIBITOR | |||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_694] | DEXFOSFOSERINE | VI4F0K069V | |||
| AMINO ACID SUBSTITUTION | [1_527] [1_542] [1_680] [1_689] [1_704] [1_790] [1_904] [1_950] | TYROSINE O-PHOSPHATE | 2R86C98KDX |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|