Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 17:24:06 GMT 2025
by
admin
on
Tue Apr 01 17:24:06 GMT 2025
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
CTZ3P20I6M
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
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| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
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CTZ3P20I6M
Created by
admin on Tue Apr 01 17:24:06 GMT 2025 , Edited by admin on Tue Apr 01 17:24:06 GMT 2025
|
PRIMARY | |||
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MAP2K1
Created by
admin on Tue Apr 01 17:24:06 GMT 2025 , Edited by admin on Tue Apr 01 17:24:06 GMT 2025
|
PRIMARY | |||
|
Q02750
Created by
admin on Tue Apr 01 17:24:06 GMT 2025 , Edited by admin on Tue Apr 01 17:24:06 GMT 2025
|
PRIMARY | |||
|
Q02750
Created by
admin on Tue Apr 01 17:24:06 GMT 2025 , Edited by admin on Tue Apr 01 17:24:06 GMT 2025
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
INHIBITOR -> TARGET |
Incorporation of [J33P]phosphate from [J33P]ATP into ERK2
UNCOMPETITIVE
IC50
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET |
IN-VITRO
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INHIBITOR -> TARGET |
IC50
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
REVERSIBLE
Ki
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_291] | THREONINE PHOSPHATE | 3L4WX7B1EI |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|