Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 16:42:40 GMT 2025
by
admin
on
Tue Apr 01 16:42:40 GMT 2025
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
PG244BS39U
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Preferred Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
PG244BS39U
Created by
admin on Tue Apr 01 16:42:40 GMT 2025 , Edited by admin on Tue Apr 01 16:42:40 GMT 2025
|
PRIMARY | |||
|
P13945
Created by
admin on Tue Apr 01 16:42:40 GMT 2025 , Edited by admin on Tue Apr 01 16:42:40 GMT 2025
|
PRIMARY | |||
|
BETA-3_ADRENERGIC_RECEPTOR
Created by
admin on Tue Apr 01 16:42:40 GMT 2025 , Edited by admin on Tue Apr 01 16:42:40 GMT 2025
|
PRIMARY | |||
|
P13945
Created by
admin on Tue Apr 01 16:42:40 GMT 2025 , Edited by admin on Tue Apr 01 16:42:40 GMT 2025
|
PRIMARY |
| From | To |
|---|---|
| 1_110 | 1_196 |
| 1_189 | 1_195 |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_8 |
| N | 1_26 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
INHIBITOR -> TARGET |
|
||
|
|
AGONIST -> TARGET |
EC50
|
||
|
RADIOLIGAND->TARGET |
Chinese hamster ovary (CHO) cells stably expressing the three ?-adrenergic receptor subtypes at comparable levels.
Kd
|
||
|
TARGET->WEAK AGONIST |
Assay in chinese hamster ovary (CHO) cells stably expressing the three ?-adrenergic receptor subtypes at comparable leve50 to 80 pM 125I-CYP were used as radioligand. Experiments were done in the presence of 100 µM GTP.
Ki
|
||
|
INHIBITOR -> TARGET |
Chinese hamster ovary (CHO) cells stably expressing the three ?-adrenergic receptor subtypes at comparable levels.
Kd
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
Assay in chinese hamster ovary (CHO) cells stably expressing the three ?-adrenergic receptor subtypes at comparable leve50
to 80 pM 125I-CYP were used as radioligand. Experiments were done in the presence of 100 µM GTP.
Ki
|
||
|
AGONIST -> TARGET |
|
||
|
AGONIST -> TARGET |
|
||
|
AGONIST -> TARGET |
SELECTIVE
|
||
|
AGONIST -> TARGET |
|
||
|
AGONIST -> TARGET |
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
|
AGONIST -> TARGET |
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
|
||
|
|
AGONIST -> TARGET |
|
||
|
|
AGONIST -> TARGET |
|
||
|
AGONIST -> TARGET |
Assay in chinese hamster ovary (CHO) cells stably expressing the three ?-adrenergic receptor subtypes at comparable leve50 to 80 pM 125I-CYP were used as radioligand. Experiments were done in the presence of 100 µM GTP.
|
||
|
|
AGONIST -> TARGET |
|
||
|
AGONIST -> TARGET |
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|
||||
| Molecular Formula | CHEMICAL |
|