Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 16:48:54 GMT 2025
by
admin
on
Tue Apr 01 16:48:54 GMT 2025
|
| Protein Type | ENZYME |
| Protein Sub Type | TYROSINE KINASE |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
RSO83C9PIA
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
|
Preferred Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
P21860
Created by
admin on Tue Apr 01 16:48:54 GMT 2025 , Edited by admin on Tue Apr 01 16:48:54 GMT 2025
|
PRIMARY | |||
|
P21860
Created by
admin on Tue Apr 01 16:48:54 GMT 2025 , Edited by admin on Tue Apr 01 16:48:54 GMT 2025
|
PRIMARY | |||
|
RSO83C9PIA
Created by
admin on Tue Apr 01 16:48:54 GMT 2025 , Edited by admin on Tue Apr 01 16:48:54 GMT 2025
|
PRIMARY |
| From | To |
|---|---|
| 1_10 | 1_37 |
| 1_137 | 1_164 |
| 1_167 | 1_175 |
| 1_171 | 1_183 |
| 1_191 | 1_199 |
| 1_195 | 1_207 |
| 1_208 | 1_216 |
| 1_212 | 1_224 |
| 1_227 | 1_236 |
| 1_240 | 1_267 |
| 1_271 | 1_282 |
| 1_286 | 1_301 |
| 1_304 | 1_308 |
| 1_481 | 1_490 |
| 1_485 | 1_498 |
| 1_501 | 1_510 |
| 1_514 | 1_530 |
| 1_533 | 1_546 |
| 1_537 | 1_554 |
| 1_557 | 1_566 |
| 1_570 | 1_591 |
| 1_594 | 1_602 |
| 1_598 | 1_610 |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_107 |
| N | 1_231 |
| N | 1_334 |
| N | 1_389 |
| N | 1_395 |
| N | 1_418 |
| N | 1_450 |
| N | 1_503 |
| N | 1_547 |
| N | 1_597 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
LIGAND->TARGET |
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|
INHIBITOR -> TARGET | |||
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|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
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|
INHIBITOR -> TARGET | |||
|
LIGAND->TARGET |
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|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
ISU104 completely suppressed Heregulin HRG-induced phosphorylation
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|
INHIBITOR -> TARGET |
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|
LIGAND->TARGET |
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|
|
INHIBITOR -> TARGET |
IgG1 bispecific antibody with enhanced antibody-dependent cell-mediated cytotoxicity (ADCC) activity targeting HER2 and HER3 receptors.
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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LIGAND->TARGET |
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INHIBITOR -> TARGET |
BINDING
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|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
|
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_667] [1_963] | DEXFOSFOSERINE | VI4F0K069V |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|