Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Mon Mar 31 23:32:04 GMT 2025
by
admin
on
Mon Mar 31 23:32:04 GMT 2025
|
| Protein Type | TRANSPORTER |
| Protein Sub Type | |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
B46KUN2O9L
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
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Common Name | English | ||
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Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
| Classification Tree | Code System | Code | ||
|---|---|---|---|---|
|
UCSF-FDA TRANSPORTAL |
SLC47A2
Created by
admin on Mon Mar 31 23:32:04 GMT 2025 , Edited by admin on Mon Mar 31 23:32:04 GMT 2025
|
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
SLC47A2
Created by
admin on Mon Mar 31 23:32:04 GMT 2025 , Edited by admin on Mon Mar 31 23:32:04 GMT 2025
|
PRIMARY | |||
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B46KUN2O9L
Created by
admin on Mon Mar 31 23:32:04 GMT 2025 , Edited by admin on Mon Mar 31 23:32:04 GMT 2025
|
PRIMARY | |||
|
Q86VL8
Created by
admin on Mon Mar 31 23:32:04 GMT 2025 , Edited by admin on Mon Mar 31 23:32:04 GMT 2025
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER |
IC50
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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SUBSTRATE -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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SUBSTRATE -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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SUBSTRATE -> TRANSPORTER |
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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SUBSTRATE -> METABOLIC ENZYME | |||
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SUBSTRATE -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> METABOLIC ENZYME | |||
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SUBSTRATE -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER |
IC50
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INHIBITOR -> TRANSPORTER | |||
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NON-SUBSTRATE -> TRANSPORTER |
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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SUBSTRATE -> TRANSPORTER | |||
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SUBSTRATE -> TRANSPORTER |
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SUBSTRATE -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER |
WEAK
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INHIBITOR -> TRANSPORTER | |||
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SUBSTRATE -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER |
corrected for non-specific binding
IC50
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER |
IN VITRO
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER |
Rifamycin is an inhibitor of renal transporters organic anion transporter (OAT) 3, multidrug and toxin extrusion (MATE) 1, and MATE2-K transporters in vitro, however, based on systemic concentrations of rifamycin observed after administration of the recommended dose, clinically relevant inhibition of these transporters in vivo is unlikely.
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER |
IC50
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INHIBITOR -> TRANSPORTER |
IC50
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SUBSTRATE -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER |
The results suggest that KLISYRI has no clinically meaningful effect on the PK of drugs mediated by MATE2-K
IC50
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INHIBITOR -> TRANSPORTER | |||
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SUBSTRATE -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER |
IC50
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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SUBSTRATE -> TRANSPORTER | |||
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SUBSTRATE -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER | |||
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INHIBITOR -> TRANSPORTER |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT:NUMBER(CALCULATED) | CHEMICAL |
|